Azetidine synthesis by La(OTf)3-catalyzed intramolecular regioselective aminolysis of cis-3,4-epoxy amines
نویسندگان
چکیده
Azetidine is a prevalent structural motif found in various biologically active compounds. In this research paper, we report La(OTf) 3 -catalyzed intramolecular regioselective aminolysis of cis -3,4-epoxy amines to afford azetidines. This reaction proceeded high yields even the presence acid-sensitive and Lewis basic functional groups.
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ژورنال
عنوان ژورنال: Frontiers in Chemistry
سال: 2023
ISSN: ['2296-2646']
DOI: https://doi.org/10.3389/fchem.2023.1251299